Cov hmoov stanozolol (winstrol) tiv thaiv cov leeg nqaij atrophy Antrophy Cas: {10418-03-8

Cov hmoov stanozolol (winstrol) tiv thaiv cov leeg nqaij atrophy Antrophy Cas: {10418-03-8
Khoom Taw qhia:
Stanozolol (Winstrol) hmoov nplej yog cov khoom siv hluavtaws Androgenic Anabolic Steroid (AAS) uas tau nyiam cov nyhuv anabolic thiab cov haujlwm tsawg. Stanozolol tau tsim thawj zaug los ntawm Winthrop lub chaw soj ntsuam nyob rau xyoo 1960 thiab yog siv los kho anemia, txhawb cov nqaij so ntswg, thiab tiv thaiv cov leeg leeg. Nws cov hmoov nyoos feem ntau yog cov xim dawb lossis tawv-dawb crystalline hmoov nrog solubility tsis tshua muaj, tab sis nws tuaj yeem coj mus rau hauv daim ntawv ntawm kev ncua lossis ntsiav tshuaj. Winstrol tuaj yeem nce cov protein ntau ntxiv, txo cov dej ua kom huv, thiab ua kom cov leeg tawv, yog li nws tau nyiam los ntawm kev ua haujlwm ntawm lub cev thiab taug qab thiab ncaws pob. Ib qho ntxiv, nws tuaj yeem txhawb nqa cov qe ntshav liab ntau thiab txhim kho kev pa oxygen muaj peev xwm, yog li ua kom muaj zog ua kom tiav thiab lub zog tawg. Txawm li cas los xij, stanozolol yog tshuaj lom rau daim siab, tshwj xeeb tshaj yog nyob rau hauv daim ntawv. Kev siv sijhawm ntev lossis cov kev siv yuav ua rau lub siab puas, cholesterolal txawv txav, thiab testosterone suprression. Yog li ntawd, nws raug nquahu kom siv nws nyob rau hauv ib qho kev ntsuas roj teeb tsim nyog thiab muaj kev tiv thaiv daim siab kom txo qis kev pheej hmoo.
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Cov khoom lag luam

 

### ** 1. Tshuaj lom neeg cov khoom thiab cov ntaub ntawv yooj yim **

** 1. Tshuaj lom neeg lub npe thiab qauv **

Stanozolol (Winstrol), lub npe luam tawm **}}}}}}}}}} c] pyrazole **. Cov mis molecular yog ** c21h32n2o **, thiab cov molecular hnyav yog ** 328.49 g / mol **.

** Tus lej lej **: ** {10418-03-8}}}}} **, yog ib cov khoom siv hluav taws xob thoob ntiaj teb siv rau kev tsim khoom thiab luam ntawm cov khoom nyoos.

** 2. Lub cev lub cev **

- ** Pom zoo ** ** (dawb lossis o-dawb crystalline hmoov.

- ** Solubility **: Soluble me ntsis hauv dej (nrog kev pab ntawm lub cosvent), yooj yim soluble hauv cov ethanol thiab chloroform.

- ** Melting point **: Txog 155-160} degree, nrog lub thermal stability ntawm cov neeg steroid sib xyaw.

- ** Qog kho qhov muag pom **: Nws yog nquag ua haujlwm, nrog kev sib hloov tshwj xeeb ntawm +36 degree rau {2}} degree (hauv ethanol).

** 3. Tshuaj lom neeg stability **

- Nws yog rhiab rau lub teeb thiab yuav tsum tau muab cia kom deb ntawm lub teeb;

- Nws yog qhov ruaj khov rau lub sijhawm ntev nyob rau hauv ib qhuav, tsawg (2-8} degree) ib nrab degree) ib nrab degree) ib nrab degree) ib nrab degree) ib nrab degree) ib nrab degree) ib nrab degree) ib nrab degree) ib nrab degree) ib nrab degree) ib nrab degree) ib nrab degree) ib nrab degree) ib nrab degree) ib nrab degree) ib nrab degree) ib nrab degree) ib nrab degree) ib nrab degree) ib puag ncig;

- Nws tuaj yeem yauv mus ua kev thaj chaw thaum raug cov kua qaub muaj zog lossis muaj zog.

 

### ** 2. Chaw muag tshuaj ua thiab kev siv hluav taws xob **

** 1. Androgenic thiab anabolic cuam tshuam **

Stanozolol siv nws cov kev cuam tshuam los ntawm kev khi rau tus ** androgen receptor (ar) **, thiab muaj ob qho tib si thiab ** cim Anabolic haujlwm **:

- ** ANABOLOLIC TXAWV **: Nws txhawb nqa cov synthesis, inhibits catabolism, thiab nce leeg nqaij;

- ** androgenic cuam tshuam **: nws tswj hwm tus txiv neej sib deev ob leeg, tab sis kev ua tsis tshua muaj (li 30% ntawm testosterone).

** 2. Anti-estrogen khoom **

- Tsis muaj kev sib txawv (tsis txhob hloov dua siab tshiab rau estrogen), zam kev phiv tshuaj estrogen-cuam tshuam xws li txiv neej lub mis loj hlob;

- Qib Testosterone ntau ntxiv los ntawm ** kev sib deev hormone bindging globulin (shebg) **.

** 3. Hematological cuam tshuam **

- Tsim kom muaj ** erythropoietin (EPO) ** Kev zais, nce cov ntshav liab suav, thiab txhim kho oxygen nqa muaj peev xwm;

- Clinically siv los kho cov tshuaj lom neeg angioedema (Hae) thiab anemia.

 

### ** 3. Thaj chaw thov **

** 1. Kev Kho Mob Siv **

- ** QIS HEREDITEMA (HEA) **: CAHE) **: Cov tsos mob los ntawm kev nce ua ke C1 esterase Inhibitors;

- ** Osteoporosis **: Txhawb pob txha ua kom nce ntxiv;

- ** Kab mob uas muaj kab kab mob uas muaj mob kas cees rau kabmob Cance): Txo cov leeg leeg.

** 2. Kev Ua Si Ua Si thiab Kev Siv Kev Ua Haujlwm ** (Tsis Yog Kev Siv Kho Mob, Ceev Faj ntawm Kev Txaus Ntseb)

- ** Kev tw kis las **: Thaum tsim txom tau tsim txom thiab ua kom muaj kev ntxhov siab (tam sim no txwv los ntawm lub ntiaj teb anti-doping lub koomhaum Wada);

- ** Daim duab Qoj Qoj Qog yog siv rau hauv cov rog poob theem kom khaws cov leeg leeg.

** 3. Daim Ntawv Thov Vaj Ntxhua Khaub Ncaws **

- ** Nees sib tw thiab dev **: txhim kho kev ua tau zoo thiab nrawm rov qab los ntawm kev raug mob;

- ** Appetite stimulant **: Siv rau kev noj zaubmov txhawb rau cov tsiaj txhu lossis tsiaj muaj mob.

 

### ** 4. Qhov tseem ceeb ntawm stanozolol **

1. ** High Anabolic / Androgenic piv **: Tus piv yog txog 320: 1, muaj cov leeg tseem ceeb tau txais cov nyhuv thiab tsawg dua Androgenic phiv.

2. ** Tsawg Hepatotoxicity ** (txheeb ze rau lwm tus {1}} Kev siv steroids luv luv): Cov khoom siv luv luv ntawm daim siab muaj nuj nqi.

3. ** Qhov ncauj thiab txhaj ntxiv daim foos DOSAGE **: APIs tuaj yeem ua tiav rau hauv cov ntsiav tshuaj lossis roj kom tau raws li cov kev xav tau sib txawv.

4. 4 Tsis muaj cov kev phiv tshuaj ntxiv **: Tsis ua rau edema lossis txiv neej lub mis.

5. ** Metabolism ceev dua **: Ib nrab-lub neej ntawm txog li 9 teev, yooj yim kho ntau npaum li cas.

 

### ** 5. Cov txheej txheem hluavtaws thiab kev tswj hwm zoo **

** 1. Synthesis txoj kev **

Kev lag luam tsim ntawm stanzolol feem ntau yog raws li ** kev hloov kho txheej txheem ntawm testosterone derivatives **:

- ** Kauj ruam tseem ceeb **:

- Qhia txog methyl pawg ({17 - alkylation) ntawm C17 txoj hauj lwm los txhim kho qhov ncauj;

- Qhia cov qauv pyrazone ntawm lub nplhaib los txhim kho teeb pom kev ruaj khov.

** 2. Tswjhwm qauv **

- ** Purity yuav tsum muaj kev coj dawb huv **: API kev coj dawb huv ntau dua los yog sib npaug rau 98% (hplc nrhiav kom pom);

- ** Kev tswj hwm tus kabmob ": suav nrog cov txheej txheem impurities (xws li siv tsis tau yam nruab nrab) thiab cov khoom lag luam (xws li oxidized impurities);

- ** Kev tshawb nrhiav txoj hauv kev **:

- ** HPLC-UV **: Qua qhov tshwj xeeb ntawm cov khoom tseem ceeb;

- ** GC-MS **: Nrhiav kom tau ntawm cov teeb meem organic;

- ** *** infrared spectroscopy (ir) **: kev pom zoo.

** 3. Cia ntawm APIIS **

- Nws yuav tsum tau muab khi thiab tiv thaiv los ntawm lub teeb, thiab cov av noo yuav tsum tau tswj hwm qis dua 40%;

- Lub saw txias ({2-8 degree) yog xav tau thaum thauj mus los tiv thaiv kev ua pa hluav taws xob.

 

### ** 6. Kev phiv thiab kev pheej hmoo **

1. ** Kev siv plawv plawv **: Siv tau ntev ntev yuav txo HDL ("cholesterol) thiab nce txoj kev pheej hmoo ntawm arteriosclerosis.

2. ** HEPATOTEXICITY **: Txawm hais tias cov koob tshuaj tiv thaiv tsawg, cov tshuaj ntau tseem tuaj yeem ua rau nce kev hloov chaw.

3. ** Kev cuam tshuam endocrine cuam tshuam **: inhibits tapogenoustosterone zais cia thiab yuav tsum tau pct (kev siv pct (post-kev voj voog).

4. "Kev ua haujlwm tsis xis nyob **: Vim tias txo cov hluavtaws collthesis, nws yuav ua rau noob tawv.

 

### ** 7. Raws li kev cai lij choj **

1. ** Kev tswj hwm thoob ntiaj teb **:

- ** WADA **: teev raws li txwv tsis pub siv hauv S1 qeb, cov kis las raug txwv tsis raug siv los ntawm kev siv nws sab hauv thiab sab nraud qhov kev ua si;

- ** USA **: DEA DESTS nws nyob rau lub sij hawm III ntawm cov tswj hwm kev ua;

- ** EU **: Nws yuav tsum tau yuav ntawm cov tshuaj noj thiab raug txwv los ntawm kev ncig ua rau cov hom phiaj tsis yog kev kho mob.

2. ** Kev cai lij choj Suav teb **:

- Raws li cov cai ntawm kev tswj hwm ntawm cov tshuaj narcotic thiab cov tshuaj psychotropic, stanog ntawm stimulants **, thiab nws yuav tsum tau kev pom zoo los ntawm xeev cov chaw noj mov thiab tshuaj noj.

 

### ** 8. Kev Lag Luam Kev Lag Luam thiab API muab saw hlau **

1. ** Lub teb chaws tsim loj **: Tuam Tshoj, Is Nrias teb, thiab Mexico yog lub ntiaj teb cov neeg xa khoom tseem ceeb;

2. ** Tus nqi hloov pauv **: Cuam tshuam los ntawm kev nruj cov cai ntawm cov cai, tus nqi lag luam hauv 2023 yog li $} / sib paub 98%);

3. "Muab cov khoom sib txuas tau sib tw **: Vim yog kev saib xyuas nruj tshaj plaws, yuav tsum muaj kev cai lij choj yuav tsum muaj kev sib raug zoo GMP kev muaj ntawv pov thawj muaj pov thawj.

 

### ** 9. Cov Lus Qhia Yav Tom Ntej **

1. ** Kev ua kom zoo nkauj ": txhim kho tsis {1}}} alkylated analogs kom txo Hepatotoxicity;

2. ** Lub kaw lus tawm tshuaj tshiab **

3. ** Kev nthuav dav qhia txog ": Tshawb xyuas nws cov kev kho mob muaj peev xwm hauv cov leeg dystrophy (xws li als).

 

### ** Ntsiab Lus **

Raws li classic anabolic steroid, stanozolol muaj cov keeb kwm keeb kwm ua haujlwm hauv ob daim teb kho mob thiab kis las. Kev tsim kho, kev tswj hwm zoo thiab kev cai lij choj ntawm nws cov ntaub ntawv raw yuav tsum ua raws thoob ntiaj teb thiab cheeb tsam cov cai. Yav tom ntej, nrog kev nkag siab tob tob ntawm cov tshuaj steroids, txhim kho cov tshuaj ntawm stanozolol yuav txo cov kev sib raug zoo thaum nthuav dav cov xwm txheej.

 

 

Txhawb nqa txoj kev them nyiaj thiab tiv tauj peb

 

Txhawb txoj kev them nyiaj
 
 

Peb txhawb ntau txoj kev them nyiaj

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Cim npe nrov: Cov hmoov stanozolol (winstrol) tiv thaiv cov leeg antrophy Cas: {} {{{{}} cov chaw tsim khoom, cov chaw tsim khoom, Hoobkas

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