Khoom Taw Qhia
Lub Npe:Ivermectin
Cov txiaj ntsig ntawm cov khoom:Haib anti-parasitic
CAS:70288-86-7
Muaj peev xwm:5 mg * 100 tabl
Daim ntawv foos:Cov ntsiav tshuaj tiav (hepius)
Txee Lub Neej:2-3Xyoo (Lub hnub ntim khoom yuav muaj yeej)
Taw qhia rau hepius hom mroupermectin
** HEPIIUS hom Irocermectin ** yog ib qho tshuaj tiv thaiv kev tiv thaiv kev siv tshuaj tua kab mob, ib yam dig muag), dej dig muag), thiab lwm yam kab mob hanthenth thiab ectoparasitic. Nws yog cov hom tshwj xeeb yog rau chav kawm tshuaj ** Ivermectin **.
### 1. ** Lub cev thiab tshuaj lom neeg **
- ** Tshuaj lub npe **: Ivermectin yog ib yam khoom ntuj tsim los ntawm **Streptomyces avermitilis**, thiab nws cov qauv muaj ntau lub nplhaib thiab ntau pawg ua haujlwm.
- **Molecular formula**: C₁₉H₃₁NO₃
* Molecular hnyav: ~ 875.56 g / mol
- ** Zoo**: Feem ntau yog dawb los yog tawm-dawb crystalline hmoov.
- ** Solubility **:
- Solubility Qes hauv dej, tab sis soluble nyob rau hauv feem ntau cov kuab tshuaj muaj ethanol, acetone, chloroform, thiab lwm yam.
- Relatively hydrophobic, yooj yim rau khi rau cov ntaub so ntswg adipose.
- ** Stability **: ruaj khov ntawm chav tsev kub, tab sis rhiab rau lub teeb thiab av noo. Tsis txhob raug ncaj qha rau lub teeb thaum lub sijhawm khaws cia ntev.
### 2. ** MECHNATORATIC THIAB TSHUAB **
Ivermectis feem ntau ua rau cov leeg ntshav ntawm cab. Nws khi rau ** -aminobutyric acid (Gaba) receptors **, nce chloride ion permeability, thiab yog li ua rau tuag tes tuag taw thiab tuag ntawm cab. Nws tseem cuam tshuam nrog ** Glutamate-gated chloride channels **, uas tseem yog tus yuam sij rau nws cov kev ua tshuaj tua kab mob.
- ** TSIS TXAUS SIAB RAU COV NEEG ": Ivermectin muaj affinity tsawg rau Gaba Receptors hauv tib neeg thiab lwm yam tsiaj muaj tsiaj, yog li nws muaj tus tswv tsev tsawg.
### 3. **Kuaj**
Qhov koob tshuaj Ivermectin feem ntau yog txiav txim los ntawm lub cev hnyav thiab hom kab mob:
- ** koob tshuaj rau cov neeg laus ib txwm muaj**: Tus qauv koob tshuaj rau kev kho mob helminthiasis muaj zog (xws li dej dig muag, lymphatic filariasis, thiab lwm yam) yog hais txog **150-200 micrograms/kg** ntawm lub cev hnyav, noj qhov ncauj raws li ib tug ib koob.
- Rau lwm yam kab mob parasitic, koob tshuaj yuav txawv.
Thov nco ntsoov tias cov koob tshuaj yuav tsum tau kho raws li tus kws kho mob cov lus qhia.
### 4. ** Ib nrab-lub neej **
Lub ** ib nrab neej ** ntawm Ivermectin yog hais txog **18-24 teev**, tab sis nws cov kev ua tau zoo feem ntau yog ntev dua, yog li nws feem ntau muab ib zaug ib zaug. Nws cov concentration hauv cov ntshav tuaj yeem maj mam txo qis dua ob peb hnub, tab sis nws cov metabolites nquag siv qee zaum tseem nyob ib ntus.
- ** Plasma ib nrab-lub neej **: txog ** 18 teev **
- **Metabolism**: Feem ntau metabolized nyob rau hauv daim siab los ntawm cytochrome P450 enzymes (tshwj xeeb tshaj yog CYP3A4), thiab metabolites raug tso tawm los ntawm cov zis thiab cov kua tsib.
### 5. ** Pharmacokinetics **
- ** Rho tawm **
- ** Kev faib tshuaj ** Cov tshuaj no tau faib tawm thoob plaws lub cev, tshwj xeeb tshaj yog hauv cov ntaub so ntswg, cov leeg, mob siab thiab lub hlwb thiab lub hlwb thiab lub hlwb thiab lub hlwb thiab lub hlwb thiab lub hlwb thiab lub hlwb thiab lub hlwb thiab lub hlwb thiab lub hlwb thiab lub hlwb.
**Metabolism thiab excretion**:
- Metabolized los ntawm daim siab, qee cov metabolites tsis muaj zog yog tsim tawm.
- Feem ntau ntawm cov tshuaj yog tawm hauv cov quav, thiab ib qho me me tawm hauv cov zis.
### 6. **Siv lub voj voog**
- ** Ib qho tshuaj rau ib leeg **: feem ntau yuav tsum muaj ib koob tshuaj.
- ** Txoj kev khomob txuas ntxiv **: Qee yam kab mob (xws li dej dig muag) yuav xav tau ntau yam kev kho mob ntawm cov sijhawm ntawm no ** {1}} lub hlis **.
### 7. **Kev qhia thiab ua tau zoo**
- ** Tus mob parasitic **:
- Dej dig muag (onchocciasis)
- Lymphatic filariasis
- muaj zog
- Neurocysticercosis
- ** Cov mob parasitic sib kis tau **:
- Qee yam kab mob parasitic tau kis los ntawm yoov tshaj cum.
- Kev kho ntshauv thiab cov kab mob.
### 8. ** Kev mob tshwm sim thiab contraindications **
- ** Cov kev mob tshwm sim ib txwm **:
- Mob taub hau me, xeev siab, poob ntawm qab los, qaug zog, thiab lwm yam.
- Cov kev mob tshwm sim tsawg dua tuaj yeem suav nrog pob khaus, lub siab ua haujlwm tsis zoo, qhov muag mob, thiab lwm yam.
- ** Cov kev phiv loj heev**: Yog tias muaj kev tsis haum tshuaj hnyav, tsis meej pem, ua pa nyuaj, lub plawv dhia tsis zoo, thiab lwm yam tshwm sim, tsum tsis txhob noj tshuaj tam sim ntawd thiab nrhiav kev pab kho mob.
** Contraindications **:
- Cov poj niam cev xeeb tub thiab pub niam mis yuav tsum siv ceev faj, tshwj xeeb tshaj yog tsis muaj kev qhia kho mob.
- Cov neeg mob uas ua xua rau Ivermectin yuav tsum zam kev siv nws.
### 9. **Kev ceev faj**
- **Kev sib cuam tshuam ntawm cov tshuaj**: Ivermectin tuaj yeem cuam tshuam nrog qee yam tshuaj, tshwj xeeb tshaj yog cov tshuaj tiv thaiv kab mob vwm (xws li phenytoin), qee yam tshuaj tiv thaiv kab mob (xws li ketoconazole), thiab lwm yam, uas tuaj yeem ua rau lawv cov tshuaj lom lossis txo lawv cov txiaj ntsig.
- ** Daim siab thiab lub raum ua haujlwm **: Rau cov neeg mob uas muaj lub siab tsis zoo thiab lub raum ua haujlwm, cov koob tshuaj yuav tsum tau hloov kho.

HEPIUS hom Ivermectin siv thiab ntau npaum li cas
HEPIUS hom Ivermectin yog cov tshuaj tiv thaiv kab mob dav siv los kho ntau yam kab mob tshwm sim los ntawm cov kab mob cab. Cov hauv qab no yog cov lus qhia ntxaws ntxaws rau cov neeg siv tshuaj, txoj hauv kev ua haujlwm, thiab kev siv thiab ntau npaum li cas:
### Cov pejxeem:
Ivermectin yog tsuas yog siv rau cov pab pawg hauv qab no:
1. ** Kev kho mob ntawm tus kab mob parasitic **:
- ** A Riven dig muag (onchociab) **: parasitic kab mob los ntawm filariasis.
- **Lymphatic Filariasis**: lymphatic system kis los ntawm filariasis.
- ** Tus kab mob cab **: Cov kab mob plab hnyuv ua rau cov kab mob sib txawv, cov hookworms, whipworms, thiab Filarial cab.
- ** Cov kiav txhab **: Kab mob kab mob los ntawm cov kiav txhab.
- ** Pediculosis capitis **: kab mob ntawm daim tawv nqaij tshwm sim los ntawm cov ntshauv.
2. **Kev tiv thaiv thiab kho cov kab mob tshwm sim los ntawm lwm yam kab mob**:
- ** QUB ANNISROSING SCHANTOSOMIAS **: Kab mob tshwm sim los ntawm Schistosomiasis.
- ** LWM YAM TSHUAJ LOS NTAWM PARASSITE **: Xws li cov kab mob qhov muag, pob ntseg pob ntseg, thiab lwm yam.
### Txoj Cai Ua Haujlwm:
Ivermectin ua haujlwm los ntawm kev cuam tshuam nrog cov kab mob hauv lub paj hlwb, tshwj xeeb tshaj yog los ntawm kev khi rau cov kab mob GABA (gamma-aminobutyric acid) receptors los inhibit paj hlwb. Qhov no tuaj yeem ua rau tuag tes tuag taw ntawm cov kab mob hauv lub paj hlwb thiab cov leeg nqaij, yog li tua cov cab lossis ua rau nws tsis muaj peev xwm txav mus los, thiab thaum kawg raug tshem tawm los ntawm lub cev tiv thaiv kab mob.
- ** Soj ntsuam kev nqis tes ua **: Ivermectin tuaj yeem khi rau cov recease hauv Gaba lub zog tswj hwm nrog tus cab lub zog thiab kev ua haujlwm tuag tes tuag taw thiab kev tuag.
- **Broad-spectrum effect**: Cov tshuaj tsis yog tsuas yog tiv thaiv kab mob hauv lub cev xwb, tab sis kuj tuaj yeem kho cov kab mob ntawm daim tawv nqaij xws li kab mob, kab mob taub hau, thiab lwm yam.
### ntau thiab kev tswj hwm:
Qhov ntau npaum thiab kev tswj hwm ntawm Ivermectin yuav txawv nyob ntawm seb hom kab mob twg, tus neeg mob hnyav thiab hnub nyoog. Cov hauv qab no yog cov kev siv ntau npaum li cas thiab kev siv tshuaj siv:
1. ** Cov neeg laus thiab menyuam yaus (qhov hnyav tshaj 15 kg) **:
- ** Diven dig muag **: Ib qho dej ntawm 200 micrograms / micrograms / Kg lub cev hnyav, feem ntau noj ib zaug.
- **Lymphatic filariasis**: Ib koob tshuaj ntawm qhov ncauj ntawm 150-200 micrograms/kg lub cev hnyav, feem ntau noj ib zaug.
- ** Kabmob **: Rau cov neeg laus thiab cov menyuam yaus uas lub cev hnyav, feem ntau 200 micrograms / kg lub cev hnyav yog noj ib zaug, thiab tuaj yeem rov ua dua raws li kws kho mob cov lus qhia.
- ** Cov ntshauv taub hau **: Cov neeg laus thiab cov menyuam yaus tuaj yeem noj 200 micrograms / kg lub cev qhov hnyav ntawm qhov ncauj, feem ntau yog ib koob.
2. ** Cov menyuam yaus (hnyav qis dua 15 kg) **:
- Cov tshuaj muab tshuaj yuav muab tau raws li lub cev hnyav, feem ntau 200 qhov hnyav thiab kev kho mob ntawm tus kws kho mob yuav tsum raug txiav txim los ntawm tus kws kho mob raws li cov neeg mob.
### Cov kev ceev faj:
- ** Cov teeb meem me me **: Cov neeg mob uas ua xua rau Ivermectin lossis lwm yam khoom xyaw yuav tsum tsis siv nws.
- ** Modrant thiab lactating poj niam **: Siv nrog kev ceev faj thiab yuav tsum tau siv raws li kev taw qhia tus kws kho mob.
- **Cov neeg mob uas muaj kab mob siab thiab lub raum tsis txaus**: Siv raws li kev qhia ntawm tus kws kho mob, kho cov koob tshuaj lossis saib xyuas cov ntsuas cuam tshuam.
- **Drug interactions**: Muaj peev xwm cuam tshuam cov tshuaj nrog qee yam tshuaj xws li lwm yam tshuaj tiv thaiv kab mob thiab tshuaj tiv thaiv kab mob vwm. Thaum siv, koj yuav tsum qhia koj tus kws kho mob txog lwm yam tshuaj uas koj noj.
### kev phiv:
Txawm hais tias Ivermectin feem ntau suav hais tias muaj kev nyab xeeb, qee cov kev mob tshwm sim tseem tshwm sim thaum siv, feem ntau yog:
- ** Daim tawv nqaij tiv thaiv **: xws li pob khaus thiab khaus.
- ** plab hnyuv **: xeev siab, ntuav, raws plab, thiab lwm yam.
- **Nervous system reactions**: xws li mob taub hau, kiv taub hau, insomnia, tsaug zog, thiab lwm yam.
Zuag qhia tag nrho, HEPIUS hom Ivermectin yog siv los kho ntau yam kab mob tshwm sim los ntawm cov kab mob cab, nrog rau cov txiaj ntsig tseem ceeb, tab sis cov koob tshuaj yuav tsum tau kho thiab saib xyuas raws li tus kws kho mob cov lus qhia thaum siv.

Qhov zoo ntawm HEPIUS hom Ivermectin
** Qhov zoo ntawm HEPIUS Hom Ivermectin **:
Ivermectin yog dav-spectrum Antiparasitic Antiparasitic cov tshuaj siv tau los kho ntau yam kab mob ntawm Ivermectis muaj nws cov cim tshwj xeeb hauv kev ua lag luam. Cov hauv qab no yog qee cov hom cim cov yam ntxwv tseem ceeb ntawm kev ua tau zoo, kev ua tau zoo, ntau lawm tshuab, thiab lwm yam.
### 1. ** Cov Qauv Zoo **
Raws li lub npe tshuaj muaj npe nrov, HEPIUS tau cog lus los tsim cov tshuaj uas ua tau raws li cov qauv zoo thoob ntiaj teb, tshwj xeeb tshaj yog ua raws li GMP (Good Manufacturing Practice) cov ntawv pov thawj uas yuav tsum tau ua thaum lub sijhawm tsim tshuaj. Txhua pawg ntawm HEPIUS ivermectin tau txais kev tswj hwm nruj, suav nrog kev tshuaj xyuas cov khoom siv raw, kev soj ntsuam cov txheej txheem tsim khoom, thiab kuaj cov khoom tiav kom ntseeg tau tias cov purity thiab kev nyab xeeb ntawm cov tshuaj.
- ** Purity thiab cov ntsiab lus ": Hepius hom Ivermectionin feem ntau muaj ntau dua kev coj dawb huv thiab cov ncauj lus tsis sib thooj los xyuas kom meej qhov siab tshaj plaws.
- ** QIB **: Los ntawm cov tshuab tswj hwm nruj zoo, hepius hom Iroermectin cov khoom muaj cov khoom lag luam siab.
### 2. **Kev ua tau zoo heev**
Ivermectin yog ib qho tshuaj tiv thaiv kab mob zoo. Los ntawm kev tsim cov koob tshuaj meej, HEPIUS hom ivermectin tuaj yeem tshem tawm cov kab mob hauv lub cev hauv lub sijhawm luv luv thiab txo cov tsos mob tshwm sim los ntawm cov kab mob cab. Nws tau pom tias muaj txiaj ntsig zoo hauv kev kho ntau yam kab mob parasitic, tshwj xeeb hauv cov hauv qab no:
- ** NematodeeGe **: xws li ankylosttomiasis, Taenia solium, schistosomiasis, thiab lwm yam.
- ** Batasites sab nraud **: Cov kab mob tawv nqaij xws li cov ntshauv taub hau xws li cov kab mob taub hau, demabies, demodex, thiab lwm yam.
- ** Ob lub qhov muag lub qhov muag pom kab mob ob lub qhov muag **: xws li cov kab mob qhov muag tau los ntawm cov kev hloov pauv hauv lub qhov muag.
HEPIUS ivermectin tseem tswj tau cov txiaj ntsig zoo tiv thaiv ntau yam kab mob parasite tiv thaiv kab mob, yog li nws yog ib qho ntawm cov tshuaj xaiv thawj zaug rau kev kho mob ntawm ntau cov kab mob parasitic.
### 3. **Broad spectrum antiparasitic effect**
Hepius Ivermectin's Anti-Parasitic Efficial Npog Ntau Hom Ntawm Cov Hom, tab sis kuj tseem tiv thaiv parasites uas tiv taus lwm cov tshuaj tiv thaiv kev tiv thaiv. Nws txwv tsis pub muaj txoj cai ntawm lub cev ua haujlwm ntawm cov cab, ua rau tus cab yuav tuag.
- ** Dav txuas ntxiv rau ntau yam parasites **: Hepius Ivermectin tsis yog siv dav hauv kev kho mob ntawm cov cab tsis tshua muaj tshuaj tiv thaiv kab mob.
### 4. **Kev ruaj ntseg siab**
HEPIUS hom ivermectin tau pom tias muaj kev phiv tsawg dua hauv kev sim tshuaj thiab siv mus ntev. Feem ntau, cov tshuaj yuav ua rau muaj kev phiv tshwm sim tsuas yog thaum noj cov koob tshuaj ntau lossis ntau dhau. Cov kev phiv tshwm sim muaj xws li mob taub hau, kiv taub hau, xeev siab, raws plab, thiab lwm yam.
- ** haum rau cov neeg laus thiab menyuam yaus hom Ivermectin yog qhov tsim nyog rau cov neeg laus (cov tshuaj muaj kev nyab xeeb raws li qhov hnyav), thiab muaj kev nyab xeeb ntau hauv qhov kev siv tshuaj ntau.
- ** QIB TOUXICITY **: Piv nrog ntau lwm cov tshuaj tiv thaiv antiparasitic, IvermectIn muaj qis qis toxicity thaum lub sij hawm muaj kev cuam tshuam tsawg dua thiab tswj tau cov kev tsis zoo thaum siv.
### 5. ** Zoo dua Bioavailability **
Hepius Ivermectin tau txais cov tshuaj kho thiab cov txheej txheem ntau lawm, ua rau nws muaj txiaj ntsig zoo hauv lub cev. Qhov no ua kom ntseeg tau tias cov khoom xyaw nquag siv tau zoo dua nqus thiab ua haujlwm, yog li kev txhim kho kev ua tau zoo.
- **Kev nqus tshuaj sai**: Cov khoom xyaw tshuaj ntawm HEPIUS Ivermectin tuaj yeem nkag mus rau hauv cov ntshav sai sai thiab ua rau muaj txiaj ntsig zoo.
- ** Ntev ib nrab-lub neej **: Ib nrab-lub neej ntawm cov tshuaj nyob hauv lub cev yog qhov tsis tshua muaj txiaj ntsig ntawm cov tshuaj thiab txo cov zaus ntawm kev tswj hwm.
### 6. * Siv dav **
Ntxiv rau kev kho cov kab mob cab hauv tib neeg, HEPIUS hom ivermectin kuj tau siv dav hauv chaw kho tsiaj los kho ntau yam kab mob cab hauv cov tsiaj, xws li cov kab mob sab hauv thiab sab nraud hauv yaj, nyuj, dev thiab lwm yam tsiaj.
- ** Kev siv ntau ntawm tib neeg thiab tsiaj txhu **: HEPIUS ivermectin yog qhov tsim nyog rau kev kho mob ntawm tib neeg cov kab mob thiab tseem tuaj yeem siv dav hauv kev kho tsiaj, nrog rau kev hloov pauv ntawm cov ntoo khaub lig.
### 7. ** Tus nqi tsim nyog thiab tus nqi tsim nyog **
HEPIUS hom ivermectin tau txais kev ntsuas tus nqi siab hauv kev ua lag luam vim nws tus nqi tsim nyog thiab cov txiaj ntsig kho tau zoo. Piv nrog rau lwm lub npe, HEPIUS ivermectin tsis cuam tshuam rau qhov zoo, thiab nws tus nqi kuj pheej yig, ua rau nws pheej yig rau ntau pawg neeg mob, tshwj xeeb tshaj yog nyob rau hauv cov teb chaws tsim, nrog rau cov ntawv thov dav dav.
### 8. ** Ntau Lawm Ntau Lawm Technology **
Hepius Cops cov txheej txheem niaj hnub, xws li thev naus laus zis high-precision synthesis thiab cov khoom siv tau zoo, kom ntseeg tau cov khoom lag luam thiab ruaj khov. Cov thev naus laus zis tau siv nyob rau hauv nws cov txheej txheem ntau lawm tsis tsuas yog ua kom cov nqi zoo, tab sis kuj muab cov neeg siv khoom nrog cov nqi sib tw ntau dua.
### 9. ** Hom koob npe nrov thiab kev txhawb nqa kev txhawb nqa **
HEPIUS hom muaj kev paub ntau yam tshuaj thiab kev siv thev naus laus zis. Nws pab neeg R & D muaj kev sib sib zog nqus tshwj xeeb hauv thaj tsam ntawm cov tshuaj tiv thaiv kab mob thiab tswj kev sib raug zoo nrog ntau lub chaw tshawb fawb thiab cov tuam txhab tshuaj thoob ntiaj teb kom ntseeg tau tias nws cov tshuaj R & D thiab kev tsim kho tshiab muaj peev xwm nyob twj ywm ntawm qib ua hauv kev lag luam.
Ib qho ntxiv, lub hom Hepius tseem muab cov kev pabcuam tom qab muag thiab kev txhawb nqa los pab cov kws kho mob thiab cov neeg mob tau txais kev kho mob zoo tshaj plaws thaum siv Ivermectin.
### Cov ntsiab lus:
Hepieve hom Ivermectin vam khom ntawm nws cov qauv tsim khoom lag luam zoo tshaj plaws, kev nyab xeeb ntau thiab tau muaj txiaj ntsig zoo thiab muaj kev sib tw pom tseeb hauv kev ua lag luam thoob ntiaj teb. Nws tsis yog tsuas yog ib qho ntawm cov tshuaj xaiv thawj zaug rau kev kho mob ntawm cov neeg ua haujlwm ntawm cov kws kho mob thiab cov neeg mob siab vim yog nws ua tau zoo.

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FAQ
Q: Dab tsi yog Hepius hom Ivermectin?
A: HEPIUS hom ivermectin yog cov tshuaj tiv thaiv kab mob siv feem ntau los kho cov kab mob uas tshwm sim los ntawm cov kab mob parasites, suav nrog onchocerciasis, dej dig muag, ntshauv, kab mob thiab lwm yam kab mob ntawm daim tawv nqaij. Nws tuaj yeem ua tiav cov txiaj ntsig kho mob los ntawm kev cuam tshuam cov kab mob hauv lub paj hlwb, ua rau tus kab mob tuag tes tuag taw thiab tuag.
Cim npe nrov: Hepius Ivermectin 5Mg CAS: {{{70288-86-7}}}} {{{{{{{} Cov neeg tsim khoom, cov chaw tsim khoom, Hoobkas

