Lub hauv paus rau phau ntawv





Cov khoom lag luam
#### 1. ** Cov qauv siv tshuaj thiab cov khoom siv pib **
** Tus tshuaj lom npe **: Trestolone acetate, tseem hu ua 7 - methyl {{1} □ ortestosterone acetate.
** Tus lej Cas **: 3764-87-2
** Cov mis molecular **: C₂₁h₂₈o₃
** Molecular hnyav **: 328.45 g / mol
** Cov qauv nta **: Ment yog qhov kev ua yeeb yam ntawm 19- nortexone), nrog lub sijhawm me me ntawm kev nqis tes ua los ntawm kev ua tiav ntawm cov cuab yeej siv hluav taws xob. Cov qauv kev coj ua no ua rau nws muaj lipophilic zoo heev, yooj yim rau khw hauv cov ntaub so ntswg thiab tso tawm qeeb.
** Lub cev nqaij daim tawv thiab tshuaj lom neeg **: Dawb rau Off-Whing Toastalline hmoov, insoluble hauv dej, yooj yim solve hauv ethanol thiab DMO. Nws yuav tsum tau muab cia kom deb ntawm lub teeb thiab ntawm qhov kub tsawg (2-8 degree) los tswj kev ruaj khov.
### 2. ** Cov yam ntxwv ua thiab ua yeeb yam **
** Receptor aquinity **: Raws li ib tug muaj zog Andrent Androgen receptor (AR) {}} Txoj kev mob sab nrauv, thiab muaj cov kev mob tshwm sim ncaj qha (xws li prostate hyperplasia).
** Holdenolic Pathway **: Nws yog hydrolyzed rau hauv cov kev nquag ua ntawm lub siab los ntawm daim siab, nrog ib nrab-lub neej ntawm {teev, uas yog qhov zoo dua li pressosterone esters. Nws cov cim kev sib tw metabolic txo qhov kev pheej hmoo ntawm Hepatotoxicity.
** Xaiv cov txiaj ntsig **: Nws muaj cov txiaj ntsig anabolic ntawm cov leeg thiab cov pob txha, cov plaub hau (pob txuv) thiab prostate, cuam tshuam cov nqaij ntswg zoo dua.
#### 3. ** Kev thov txais kev kho mob thiab kev tshawb fawb paub **
- ** Dua **: Cov kev sim kho mob tau qhia tias muaj peev xwm txhim kho kom muaj kev sib deev ntawm cov ntshav testosterone, thiab tsis ua rau cov qe ntshav liab heev.
- ** Kev tswj cov tshuaj tiv thaiv me me li qub?
- ** HIV-RELELELE Wasting syndrome **: Rau cov leeg atrophy, kawm muaj cov txiaj ntsig anabolic zoo thiab tsis nce cov hlab ntsha muaj kev pheej hmoo.
- ** Hla kev sib deev Hormone Kev Kho Mob **: Kev tshawb fawb tshawb nrhiav nws lub peev xwm los hloov tes los ntawm poj niam ua txiv neej kev kho mob, vim nws cov kev mob tshwm sim hauv zos thiab qhov kev mob tshwm sim tsawg.
#### 4. ** Cov ntsiab lus zoo thiab muaj peev xwm sib tw **
- ** High Efficiency **: A Ua kom muaj kev ua haujlwm zoo yog 10 lub sij hawm uas ntawm Testosterone, thiab nws tuaj yeem ua tau zoo ntawm koob tshuaj tiv thaiv qis, txo qhov ntau ntawm cov tshuaj.
- ** Kev Nyab Xeeb ** Tsis txhob {5 -} {} {{1} {} {} recuctase vam khom, txo qhov kev pheej hmoo ntawm prostate hyperplasia thiab cov plaub hau poob; Tsawg daim siab muaj txiaj ntsig, haum rau kev siv ntev.
- ** Metabolic tau zoo dua **: Cov qauv tshuaj ntxiv rau lub neej ib nrab-lub neej, txhawb 1-2} lub lim tiam, thiab txhim kho cov neeg mob ua raws.
- ** GENDER-TSHWJ XEEB DAIM NTAWV THOV HAUJ LWM **: Kev tawg ua ntu zus hauv kev tiv thaiv kev tiv thaiv tus txiv neej yuav rov sau cov qauv kev ua lag luam.
### 5. ** Cov txheej txheem synthesis thiab kev tswj hwm zoo **
** Txoj kev hluavtaws synthesis **: siv estradiol raws li qhov pib, {{}}} Methyl cov tshuaj, thiab thaum kawg Esterification yog tau txais kom tau acetate. Cov kauj ruam tseem ceeb suav nrog kev tswj cov seroselective kom ntseeg tau tias 7 kev teeb tsa.
** Cov Qauv Tswj Qauv Zoo **:
- ** Purity **: HPLC nrhiav tau ntau dua lossis sib npaug nrog 99%, lub ntsiab tseem ceeb yog deycetylated (tsawg dua los yog sib npaug rau {2}}. 5%).
- ** Muab cov qauv ntawm Iich Q3c, ua tau zoo, methanol thiab ethyl acetate cov seem yog tsawg dua lossis sib luag rau 3000ppm thiab 5000ppm
- ** TSIB cov khoom siv microbial yuav tsum tau tshawb xyuas los ntawm membrane pom, endotoxin<0.2 EU/mg.
### 6. ** Raws li kev ua lag luam thiab muab cov saw hlau xa tawm **
** Muab cov chaw muag khoom tseem ceeb **:
- ** Staleroids Inc. **
- ** HOOTI LOOT ROJNZ BUCK ** (Suav Teb): Kev siv-qib khoom noj khoom haus, hais ntawm $} / g, purity ntau dua los yog sib npaug ntawm 98%.
- ** EUROPE Cov txheeb xyuas sab Europe **: Muaj los ntawm cov neeg faib khoom xws li LGC qauv, nrog tus nqi them ntawm 30% {{%.
** Kev thov ua lag luam **: Txwv los ntawm kev kuaj mob theem xwm txheej, qhov tam sim no tau xav txog cov chaw tshawb fawb thiab cov chaw thov R & DUA R &CE}}}% tom qab kev pom zoo.
#### 7. ** Kev nyab xeeb thiab cov nyom tshwm sim **
- ** Cov kev cuam tshuam tshwm sim tshwm sim **: Kev txhaj tshuaj tiv thaiv (mob, liab thiab pob txuv), muaj kev sib deev ntawm kev sib txawv ntawm<10%.
- ** Qhov txaus ntshai heev **: Cov koob tshuaj ntau heev yuav ua rau muaj kev ntseeg siab (sab nraud 1.2%), tab sis qis dua li ib txwm muaj Aas.
- ** Cov kab mob me me **: Prostate cancer, prostate cancer, mob cancer mis, mob siab rau lub siab thiab raum tsis sib xws. Yuav tsum tau saib xyuas hematocrit thiab PSA qib yuav tsum tau ua.
#### 8. ** Kev cai thiab kev ua raws li **
- ** Tebchaws Asmeskas: Tsis tau muaj npe teev tseg raws li kev tswj hwm los ntawm DEA, tab sis raws li kev tshawb fawb compound, nws yuav tsum ua raws li 21 CFR Ntu 312 (tsis raws cai).
- ** EU **: suav nrog hauv "cov ntaub ntawv tshuaj raw" cov catalog, import thiab export yuav tsum tau muab ntawv pov thawj rau Edmf.
- ** Suav **: Tsis muaj npe nyob rau hauv "kev cai ntawm kev tswj hwm ntawm cov tshuaj tsis zoo thiab tshuaj yeeb tshuaj", tab sis kev tsim cov yeeb tshuaj tsim nyog ".
#### 9. ** Cov kev sib tw yav tom ntej thiab kev sib tw **
- ** Kev kho kom haum xeeb kev kho mob **: Tshawb nrhiav kev sib xyaw nrog GNRH analogs kom txhim kho cov pab me me, lossis sib txuas nrog cov lus sib txuas los txo cov pob txha xiam.
- ** Kev txhaj tshuaj tshiab tshiab **: Kev Txhaj Tshuaj Tshiab (ib hlis ib zaug) thiab hloov pauv thaj ua rau muaj kev txhim kho cov tshuaj kom ua tau zoo.
- ** ** QICATE teeb **: PATA ntawm cov tseem ceeb tau tas sij hawm, tab sis kev sib tw rau cov txheej txheem tsim qauv (xws li kev sib tw thev naus laus zis) thiab kev ntsuas tshiab patents yog tsiv heev.
#### xaus
Ment (tritorone acetate) yuav tsum qhib txoj kev tshiab hauv thaj chaw hormones nrog nws cov khoom lag luam tshwj xeeb thiab kev kho mob. Nrog kev nce qib ntawm theem III chaw kuaj mob thiab pib ua lag luam, nws yog qhov tsim nyog tso tawm, tab sis nws yog ib qho tsim nyog los them sai sai cov ntaub ntawv kev nyab xeeb thiab cov qauv kev tswj hwm. API Cov neeg muab khoom siv yuav tsum npaj GMP ntau lawm ua haujlwm ua ntej kom tau raws li yav tom ntej loj loj ntau lawm kev xav tau.
Txhawb nqa txoj kev them nyiaj thiab tiv tauj peb
Txhawb txoj kev them nyiaj
Peb txhawb ntau txoj kev them nyiaj





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Cim npe nrov: Cov hmoov nplej sawv (trestolone acetate) tseem ceeb}}}}}} cov chaw tsim khoom, cov chaw tsim khoom, Hoobkas
